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Neurokinin receptor antagonists
Neurokinin receptor antagonists
Cyclic urea derivatives as potent NK1 selective antagonists
Organic Chemistry / Macromolecular X-Ray Crystallography / Animals / Urea / Fluorine / Rats / Bioorganic and medicinal Chemistry / Structure activity Relationship / Protein Binding / Biological Availability / Heterocyclic compounds / Molecular Structure / Neurokinin receptor antagonists / Motor activity / Rats / Bioorganic and medicinal Chemistry / Structure activity Relationship / Protein Binding / Biological Availability / Heterocyclic compounds / Molecular Structure / Neurokinin receptor antagonists / Motor activity
Cyclic urea derivatives as potent NK1 selective antagonists
Organic Chemistry / Macromolecular X-Ray Crystallography / Animals / Urea / Fluorine / Rats / Bioorganic and medicinal Chemistry / Structure activity Relationship / Protein Binding / Biological Availability / Heterocyclic compounds / Molecular Structure / Neurokinin receptor antagonists / Motor activity / Rats / Bioorganic and medicinal Chemistry / Structure activity Relationship / Protein Binding / Biological Availability / Heterocyclic compounds / Molecular Structure / Neurokinin receptor antagonists / Motor activity
Biphenyl derivatives as novel dual NK1/NK2-receptor antagonists
Organic Chemistry / Humans / Animals / Conformational Analysis / Molecular Conformation / Bioorganic and medicinal Chemistry / Biological activity / Structure activity Relationship / Molecular Structure / Neurokinin receptor antagonists / Bioorganic and medicinal Chemistry / Biological activity / Structure activity Relationship / Molecular Structure / Neurokinin receptor antagonists
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